What is a Flumazenil? For Flumazenil, many people may not know a lot about fluorine marcie is a kind of pharmaceutical raw materials, the following will introduce for you:
Flumazenil for white or white crystalline powder; Odourless and tasteless. Easily dissolved in chloroform or glacial acetic acid, slightly in methanol solution, almost insoluble in water. Benzodiazepines drugs poisoning rescue. Can also be used for the rescue of alcohol poisoning.
Flumazenil for selective medicine benzodiazepines antagonism. Its chemical structure and benzodiazepines approximation, the role of the central zhuo benzodiazepine receptors (BZD), without BZD sample blocks receptors. Animal experiments proved that it can be reversed on the central BZD receptor affinity of BZD classes and class of BZD (e.g., zopiclone, etc), to the person's role is consistent. It can also partly antagonism the anticonvulsive effect of valproic acid sodium. Antidepressant drugs can increase the secretion of prolactin level, human body and BZD anti-anxiety drugs can make it lower, the product reduce the effect of BZD class can antagonism. Of diazepam, lorazepam and triazolam and tolerability of body depend on animals, the use of this product have can produce withdrawal symptoms. This product is a weak alkali lipotropy, plasma protein combined rate at about 50%, and albumin.
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